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CETIRIZINE HYDROCHLORIDE SYRUP For Oral Use Rx only


DESCRIPTION


CLINICAL PHARMACOLOGY


Mechanism of Actions


Pharmacokinetics


Distribution


Metabolism


Elimination


Interaction Studies


Special Populations


Effect of Gender


Effect of Race


Pharmacodynamics


Clinical Studies


INDICATIONS AND USAGE


Perennial Allergic Rhinitis


Chronic Urticaria


CONTRAINDICATIONS


PRECAUTIONS


Activities Requiring Mental Alertness


Drug-Drug Interactions


Carcinogenesis, Mutagenesis and Impairment of Fertility


Pediatric Use


ADVERSE REACTIONS

   Headache 12.3%11.0%14.0%
   Pharyngitis 2.9%6.2%2.8%
   Abdominal pain 1.9%4.4%5.6%
   Coughing 3.9%4.4%2.8%
   Somnolence 1.3%1.9%4.2%
   Diarrhea 1.3%3.1%1.9%
   Epistaxis 2.9%3.7%1.9%
   Bronchospasm 1.9%3.1%1.9%
   Nausea 1.9%1.9%2.8%
   Vomiting 1.0%2.5%2.3%

Autonomic Nervous System


Cardiovascular


Central and Peripheral Nervous Systems


Gastrointestinal


Genitourinary


Hearing and Vestibular


Metabolic/Nutritional


Musculoskeletal


Psychiatric


Respiratory System


Reproductive


Reticuloendothelial


Skin


Special Senses


Vision


Body as a Whole

Occasional instances of transient, reversible hepatic transaminase elevations have occurred during cetirizine therapy. Hepatitis with significant transaminase elevation and elevated bilirubin in association with the use of cetirizine hydrochloride has been reported.


Post-Marketing Experience


DRUG ABUSE AND DEPENDENCE


OVERDOSAGE


DOSAGE AND ADMINISTRATION


Children 2 to 5 Years for Chronic Urticaria


Children 6 months to <2 years for Perennial Allergic Rhinitis and Chronic Uriticaria


HOW SUPPLIED


PACKAGE LABEL.PRINCIPAL DISPLAY PANEL